Does it upregulate or downregulate GABA(A) receptors over time? I've seen user experiences citing sedative-like properties, which makes me wonder whether it's actually a GABA agonist.
What are your experiences with this?
Posted 27 December 2012 - 11:03 PM
Posted 27 December 2012 - 11:26 PM
Posted 28 December 2012 - 09:16 AM
Posted 28 December 2012 - 10:01 AM
Edited by Raza, 28 December 2012 - 10:02 AM.
Posted 28 December 2012 - 06:04 PM
Posted 28 December 2012 - 10:26 PM
it is an opioid agonist so id say it down regulates, but I am unsure of its antagonistic activities.
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